MP-2001

MP-2001
Identifiers
  • (8R,9S,13S,14S,17S)-2,3,4-Trimethoxy-13-methyl-6,7,8,9,11,12,14,15,16,17-decahydrocyclopenta[a]phenanthren-17-ol
CAS Number
PubChem CID
ChemSpider
UNII
CompTox Dashboard (EPA)
Chemical and physical data
FormulaC21H30O4
Molar mass346.467 g·mol−1
3D model (JSmol)
  • C[C@]12CC[C@H]3[C@H]([C@@H]1CC[C@@H]2O)CCC4=C(C(=C(C=C34)OC)OC)OC
  • InChI=1S/C21H30O4/c1-21-10-9-12-13(16(21)7-8-18(21)22)5-6-14-15(12)11-17(23-2)20(25-4)19(14)24-3/h11-13,16,18,22H,5-10H2,1-4H3/t12-,13+,16-,18-,21-/m0/s1
  • Key:HRVXCJHYWIFSOQ-LEZVPBBQSA-N

MP-2001, also known as 2,3,4-trimethoxyestra-1,3,5(10)-trien-17β-ol or 2,4-dimethoxyestradiol 3-methyl ether, is a steroid and derivative of estradiol that was described in 1966 and is devoid of estrogenic activity but produces potent analgesic effects in animals. It was never marketed.

See also

References

  1. 1 2 J. Elks (14 November 2014). The Dictionary of Drugs: Chemical Data: Chemical Data, Structures and Bibliographies. Springer. p. 1248. ISBN 978-1-4757-2085-3.
  2. ↑ Axelrod LR, Baeder DH (1966). "A steroidal analgesic". Proc. Soc. Exp. Biol. Med. 121 (4): 1184–7. doi:10.3181/00379727-121-31000. PMID 5937726. S2CID 41902501.